4SC-202 tosylate ( 4SC-202 )

产品货号. M17177 CAS No. 1186222-89-8

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

4SC-202 tosylate
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
产品描述

4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
同义词

4SC-202
通路

Metabolic Enzyme/Protease
靶点

Phosphatase
受体

HDAC1;HDAC2;HDAC3;HDAC5;HDAC9;HDAC10;HDAC11;
研究领域

Cancer
适应症

——

CAS Number

1186222-89-8
分子量

619.71
分子式

C30H29N5O6S2
纯度

98%
溶解度

DMSO : ≥ 51 mg/mL. 82.30 mM
SMILES

CC1=CC=C(C=C1)S(=O)(=O)O.CN1C=C(C=N1)C2=CC=C(C=C2)S(=O)(=O)N3C=CC(=C3)/C=C/C(=O)NC4=CC=CC=C4N
化学全称

——

1. Pinkerneil M, Hoffmann M J, Kohlhof H, et al. Targeted Oncology, 2016, 11(6):783-798.

计算器

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